Generating 3D Molecules for Target Protein Binding

Authors: Meng Liu, Youzhi Luo, Kanji Uchino, Koji Maruhashi, Shuiwang Ji

ICML 2022 | Conference PDF | Archive PDF | Plain Text | LLM Run Details

Reproducibility Variable Result LLM Response
Research Type Experimental Experiments demonstrate that our Graph BP is effective to generate 3D molecules with binding ability to target protein binding sites. Our implementation is available at https://github.com/divelab/Graph BP.
Researcher Affiliation Collaboration 1Department of Computer Science & Engineering, Texas A&M University, TX, USA 2Fujitsu Research of America, INC., CA, USA 3Fujitsu Research, Fujitsu Limited, Kanagawa, Japan.
Pseudocode No The paper does not contain any pseudocode or clearly labeled algorithm blocks.
Open Source Code Yes Our implementation is available at https://github.com/divelab/Graph BP.
Open Datasets Yes We use the Cross Docked2020 dataset (Francoeur et al., 2020), which contains over 22 million docked proteinligand crystal structures, to evaluate Graph BP for structure-based drug design.
Dataset Splits No The paper mentions 'training set' and 'test set' but does not explicitly state a 'validation set' or 'validation split'.
Hardware Specification No The paper mentions 'insufficient memory budget' as a reason for not using more advanced GNNs, but it does not specify any particular hardware (e.g., GPU models, CPU types, or cloud instances) used for the experiments.
Software Dependencies No The paper mentions software like 'RDkit', 'Open Babel', 'gnina', and 'PyTorch' (implicitly), but it does not provide specific version numbers for any of these software components.
Experiment Setup No The paper mentions 'stochastic gradient descent' for training and the general architecture, but it does not provide specific hyperparameters (e.g., learning rate, batch size, number of epochs) or detailed system-level training settings.